SCHEMBL14715513

SCHEMBL14715513

CC(C)Oc1ccc2nc(N3CCC(Cc4ccccc4)(OC(=O)NCc4ccccc4)CC3)nc(O)c2c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
RAB9A P51151 1/20 0.41
THRB P10828 1/20 0.40
TP53 P04637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
ACHE P22303 2/20 0.38
RET P07949 2/20 0.38
KDM4E B2RXH2 2/20 0.37
HTR2A P28223 1/20 0.37
DRD3 P35462 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
MAPT P10636 2/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SLC2A1 P11166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715414 0.94 NPC1 (0.41) NPC1RAB9ATHRBTP53RXFP1
SCHEMBL14715298 0.88 WHR1 (0.44)
SCHEMBL14715442 0.88 WHR1 (0.44)
SCHEMBL2171045 0.87 TP53 (0.44) NPC1RAB9ATHRBTP53RXFP1
SCHEMBL14715474 0.86 MCHR1 (0.36) ACHERETKDM4EHTR2ADRD3
SCHEMBL14715274 0.86 TACR3 (0.45) RETHTR2ASLC2A1
SCHEMBL14715376 0.85 WHR1 (0.46)
SCHEMBL14715403 0.83 WHR1 (0.41) RET
SCHEMBL14715358 0.82 MCHR1 (0.42) HTR2ADRD3
SCHEMBL14715369 0.82 PDE5A (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed