SCHEMBL14715734

SCHEMBL14715734

COCCC(=O)NC1CCC(CCN2CCC(Oc3c(Cl)cc(F)cc3Cl)CC2)CC1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 20/20 0.61
HTR2A P28223 17/20 0.61
DRD2 P14416 15/20 0.61
HTR1A P08908 4/20 0.61
DRD4 P21917 4/20 0.61
HTR2B P41595 4/20 0.61
HTR2C P28335 3/20 0.61
DRD1 P21728 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3084894 1.00 DRD3 (0.61) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL3067778 0.90 DRD3 (0.61) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL3093417 0.90 DRD3 (0.61) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL3069391 0.88 DRD3 (0.51) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL14715617 0.88 DRD3 (0.51) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL3080642 0.85 DRD3 (0.61) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL14715626 0.85 DRD3 (0.61) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL14715634 0.85 DRD3 (0.45) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL3082089 0.83 DRD3 (0.55) DRD3HTR2ADRD2HTR1A
SCHEMBL230475 0.82 DRD3 (0.60) DRD3HTR2ADRD2HTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed