SCHEMBL14720745

SCHEMBL14720745

OC1(c2ccc(C=C3CCN(C4CCC4)CC3)c(Cl)c2)CCOCC1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 11/20 0.39
PDE2A O00408 2/20 0.37
PDE10A Q9Y233 2/20 0.37
OPRM1 P35372 2/20 0.37
OPRD1 P41143 2/20 0.37
OPRL1 P41146 2/20 0.37
TACR1 P25103 1/20 0.35
HTR1D P28221 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14721030 0.85 CCR1 (0.37) CCR1OPRM1OPRD1OPRL1HTR1D
SCHEMBL14720746 0.82 HRH3 (0.38) CCR1OPRL1
SCHEMBL14720847 0.80 HRH3 (0.38) CCR1OPRM1OPRL1
SCHEMBL14720603 0.79 HRH3 (0.36) CCR1OPRL1
SCHEMBL14720966 0.79 HRH3 (0.36) CCR1OPRL1
SCHEMBL14720807 0.79 HRH3 (0.36) CCR1OPRL1
SCHEMBL14720602 0.79 HRH3 (0.36) CCR1OPRL1
SCHEMBL14720811 0.77 HRH3 (0.36) CCR1OPRM1OPRL1
SCHEMBL14720813 0.77 HRH3 (0.36) CCR1OPRM1OPRL1
SCHEMBL14721107 0.77 HRH3 (0.36) CCR1OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO claimed