SCHEMBL14723667

SCHEMBL14723667

CN1CCC(COCc2cc(-c3ccncc3)cc(C(C)(F)F)c2)(c2ccccc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.67
SLC6A4 P31645 6/20 0.67
KCNH2 Q12809 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3591447 0.93 TACR1 (0.77) TACR1SLC6A4KCNH2
SCHEMBL14723659 0.88 TACR1 (0.65) TACR1SLC6A4
SCHEMBL13404228 0.83 TACR1 (0.80) TACR1SLC6A4
SCHEMBL13404225 0.82 TACR1 (0.78) TACR1SLC6A4KCNH2
SCHEMBL13404226 0.81 TACR1 (0.77) TACR1SLC6A4
SCHEMBL14723663 0.81 TACR1 (0.61) TACR1SLC6A4KCNH2
SCHEMBL1388284 0.81 TACR1 (1.00) TACR1SLC6A4KCNH2
SCHEMBL3590589 0.80 TACR1 (0.84) TACR1SLC6A4KCNH2
SCHEMBL3599336 0.80 TACR1 (0.77) TACR1SLC6A4
SCHEMBL3599901 0.80 TACR1 (1.00) TACR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8383821-B2 NK-1 and serotonin transporter inhibitors BRISTOL-MEYERS SQUIBB COMPANY (US) 2013-02-26 US disclosed