SCHEMBL14723671

SCHEMBL14723671

Fc1ccc(Cl)c(-c2cc(COCC3(c4ccccc4)CCNCC3)cc(C(F)(F)F)c2)c1

nearest known ligand 0.83

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.70
SLC6A4 P31645 2/20 0.70
KCNH2 Q12809 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13404183 0.92 TACR1 (0.74) TACR1SLC6A4KCNH2
SCHEMBL13404182 0.91 TACR1 (0.72) TACR1SLC6A4KCNH2
SCHEMBL13404119 0.91 TACR1 (0.75) TACR1SLC6A4KCNH2
SCHEMBL13404157 0.89 TACR1 (0.72) TACR1SLC6A4
SCHEMBL13404188 0.88 TACR1 (0.67) TACR1SLC6A4
SCHEMBL13404177 0.87 TACR1 (0.66) TACR1SLC6A4KCNH2
SCHEMBL13404053 0.87 TACR1 (0.66) TACR1SLC6A4KCNH2
SCHEMBL13404088 0.87 TACR1 (0.80) TACR1SLC6A4
SCHEMBL13404122 0.86 TACR1 (0.74) TACR1SLC6A4KCNH2
SCHEMBL13404136 0.86 TACR1 (0.74) TACR1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8383821-B2 NK-1 and serotonin transporter inhibitors BRISTOL-MEYERS SQUIBB COMPANY (US) 2013-02-26 US disclosed