SCHEMBL14723965

SCHEMBL14723965

Cn1c(C(=O)N2CCC(NCc3ccccc3)(C(N)=O)CC2)cc(-c2ccccc2CI)c1-c1ccc(OCCO)cc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.35
DRD2 P14416 2/20 0.34
HTR7 P34969 2/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
DRD3 P35462 1/20 0.34
HTR1A P08908 1/20 0.34
HTR6 P50406 1/20 0.34
CNR2 P34972 1/20 0.33
LTA4H P09960 2/20 0.33
NPC1 O15118 1/20 0.33
CYP46A1 Q9Y6A2 1/20 0.32
KMT2A Q03164 1/20 0.32
ADORA2B P29275 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP2D6 P10635 1/20 0.31
TP53 P04637 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12602474 0.92 CNR1 (0.35) CNR1DRD2HTR7KCNH2HRH3
SCHEMBL1128273 0.90 CNR1 (0.43) CNR1DRD2HTR7KCNH2HRH3
SCHEMBL1985069 0.87 CNR1 (0.42) CNR1KCNH2HRH3CNR2
SCHEMBL1987339 0.85 CNR1 (0.41) CNR1DRD2HTR7KCNH2HTR1A
SCHEMBL1128022 0.83 CNR1 (0.40) CNR1HTR1ACNR2ALDH1A1
SCHEMBL1127694 0.82 CNR1 (0.40) CNR1DRD2HTR7KCNH2HRH3
SCHEMBL1987361 0.81 CNR1 (0.40) CNR1HTR1ACNR2
SCHEMBL1988692 0.80 CNR1 (0.46) CNR1HTR1ACNR2
SCHEMBL1990962 0.80 CNR1 (0.42) CNR1HTR1ACNR2ALDH1A1
SCHEMBL1985030 0.77 CNR1 (0.41) CNR1KCNH2HTR1ACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8383666-B2 Pyrrole derivatives, preparation of same and therapeutic application thereof SANOFI (FR) 2013-02-26 US disclosed