SCHEMBL14726358

SCHEMBL14726358

O=C1OCc2c1ccc([C@H]1CO1)c2C1CC1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 18/20 0.46
PDE4D Q08499 1/20 0.36
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286516 1.00 KCNJ1 (0.46) KCNJ1PDE4DKCNH2
SCHEMBL29195553 0.90 KCNJ1 (0.41) KCNJ1PDE4DKCNH2
SCHEMBL2891319 0.80 KCNJ1 (0.55) KCNJ1KCNH2
SCHEMBL286208 0.80 KCNJ1 (0.55) KCNJ1KCNH2
SCHEMBL30444525 0.80 KCNJ1 (0.55) KCNJ1KCNH2
SCHEMBL30444657 0.80 KCNJ1 (0.55) KCNJ1KCNH2
SCHEMBL2899747 0.80 KCNJ1 (0.55) KCNJ1KCNH2
SCHEMBL14726115 0.79 KCNJ1 (0.53) KCNJ1
SCHEMBL286489 0.78 KCNJ1 (0.40) KCNJ1
SCHEMBL287079 0.78 KCNJ1 (0.47) KCNJ1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2744499-B1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME (US) 2016-09-28 EP disclosed
WO-2013028474-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2013-02-28 WO disclosed