SCHEMBL14726864

SCHEMBL14726864

Cc1nc(NCc2cnn(C)c2)cc(OC[C@H]2CC2c2ccc(CF)cn2)n1

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 20/20 0.82
SSTR2 P30874 1/20 0.55
KCNH2 Q12809 1/20 0.55
NR1I2 O75469 1/20 0.53
CYP2C9 P11712 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720951 1.00 PDE10A (0.82) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL15945392 1.00 PDE10A (0.82) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL14721189 0.90 PDE10A (0.84) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL14722815 0.90 PDE10A (0.84) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL14723429 0.90 PDE10A (1.00) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL14723037 0.90 PDE10A (1.00) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL14721277 0.90 PDE10A (1.00) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL14726822 0.90 PDE10A (1.00) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL14726816 0.88 PDE10A (0.80) PDE10ASSTR2KCNH2NR1I2CYP2C9
SCHEMBL14722970 0.88 PDE10A (0.80) PDE10ASSTR2KCNH2NR1I2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013028590-A1 PYRIMIDINE PDE10 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-02-28 WO disclosed