SCHEMBL14748263

SCHEMBL14748263

C[C@H]1CC[C@H](CCN2CCN(c3noc4cc(F)ccc34)CC2)CC1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 17/20 0.56
DRD2 P14416 6/20 0.56
HTR1A P08908 2/20 0.56
HTR7 P34969 2/20 0.53
DRD3 P35462 12/20 0.52
KCNH2 Q12809 1/20 0.50
SLC6A4 P31645 1/20 0.49
ACHE P22303 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13013944 0.89 HTR2A (0.56) HTR2ADRD2HTR1AHTR7DRD3
Hydrochloric Acid SCHEMBL1970211 0.88 HTR2A (0.55) HTR2ADRD2HTR1AHTR7DRD3
Hydrochloric Acid SCHEMBL1970209 0.88 HTR2A (0.55) HTR2ADRD2HTR1AHTR7DRD3
SCHEMBL14748241 0.87 HTR2A (0.52) HTR2AHTR1ADRD3
SCHEMBL14748258 0.87 HTR2A (0.51) HTR2ADRD2HTR1AHTR7DRD3
SCHEMBL22302917 0.85 HTR2A (0.53) HTR2ADRD2HTR1AHTR7DRD3
SCHEMBL12631894 0.84 HTR2A (0.54) HTR2ADRD2HTR1AHTR7
SCHEMBL12631926 0.84 HTR2A (0.54) HTR2ADRD2HTR1AHTR7
SCHEMBL22303281 0.84 HTR2A (0.54) HTR2ADRD2HTR1AHTR7DRD3
SCHEMBL21026108 0.82 DRD3 (0.61) HTR2ADRD2HTR1ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334657-B1 PIPERAZINE D3 AND 5-HT2A RECEPTOR MODULATORS HOFFMANN LA ROCHE (CH) 2013-03-06 EP disclosed