SCHEMBL14748427

SCHEMBL14748427

COc1ccc(C#N)c(Oc2ccc(B3OC(C)(C)C(C)(C)P3)c(C=O)c2)n1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.35
PDE4A P27815 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
GPR119 Q8TDV5 1/20 0.31
ERN1 O75460 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14748430 0.93 PDE4B (0.38) PDE4BPDE4APDE4CPDE4D
SCHEMBL2528076 0.86 PDE4B (0.39) PDE4BPDE4APDE4CPDE4DCYP1A2
SCHEMBL2532071 0.79 PDE4B (0.43) PDE4BPDE4APDE4CPDE4DCYP1A2
SCHEMBL2528121 0.75 CYP1A2 (0.38) PDE4BPDE4APDE4CPDE4DCYP1A2
SCHEMBL2230030 0.73 PDE4B (0.47) PDE4BPDE4APDE4CPDE4D
SCHEMBL15012608 0.72 PDE4B (0.41) PDE4BPDE4APDE4CPDE4D
SCHEMBL2230578 0.70 PDE4B (0.41) PDE4BPDE4APDE4CPDE4D
SCHEMBL2527442 0.70 PDE4B (0.44) PDE4BPDE4APDE4CPDE4D
SCHEMBL2525481 0.70 FGFR4 (0.36) PDE4BPDE4APDE4CPDE4D
SCHEMBL2528977 0.69 PDE4B (0.37) PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2564857-A1 Boron-containing small molecules as anti-inflammatory agents Anacor Pharmaceuticals, Inc. (US) 2013-03-06 EP disclosed