SCHEMBL14751306

SCHEMBL14751306

CC(C)(C)NC(=O)c1cn(COCC[Si](C)(C)C)c2ncc(-c3nn(CCCN4CC(N)C4)c4ccc(OC(F)F)cc34)nc12

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SYK P43405 18/20 0.60
KCNH2 Q12809 6/20 0.60
CYP2C9 P11712 3/20 0.60
CYP2D6 P10635 3/20 0.55
DGAT1 O75907 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14739279 0.96 SYK (0.60) SYKKCNH2CYP2C9CYP2D6DGAT1
SCHEMBL14737183 0.94 SYK (0.70) SYKKCNH2CYP2C9CYP2D6
SCHEMBL14737668 0.92 SYK (0.58) SYKKCNH2CYP2C9CYP2D6DGAT1
SCHEMBL14737822 0.92 SYK (0.70) SYKKCNH2CYP2C9CYP2D6
SCHEMBL14737571 0.91 SYK (0.57) SYKKCNH2CYP2C9CYP2D6DGAT1
SCHEMBL14737101 0.90 SYK (0.56) SYKKCNH2CYP2C9CYP2D6DGAT1
SCHEMBL14738744 0.90 SYK (0.56) SYKKCNH2CYP2C9CYP2D6DGAT1
SCHEMBL14737542 0.90 SYK (0.58) SYKKCNH2CYP2C9CYP2D6DGAT1
SCHEMBL14737786 0.90 SYK (0.68) SYKKCNH2CYP2C9CYP2D6DGAT1
SCHEMBL14737428 0.90 SYK (0.56) SYKKCNH2CYP2C9CYP2D6DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013030138-A1 PYRROLOPYRAZINE KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2013-03-07 WO disclosed