SCHEMBL14765128

SCHEMBL14765128

COc1c(Br)ccc2nc(C)c(=O)[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 3/20 0.42
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
GRIN2D O15399 3/20 0.37
GRIN3B O60391 3/20 0.37
GRIN1 Q05586 3/20 0.37
GRIN2A Q12879 3/20 0.37
GRIN2B Q13224 3/20 0.37
GRIN2C Q14957 3/20 0.37
GRIN3A Q8TCU5 3/20 0.37
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TYMS P04818 3/20 0.35
CASP3 P42574 1/20 0.33
KMT2A Q03164 2/20 0.32
MAPT P10636 1/20 0.32
DAO P14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24157397 0.81 DAO (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL30212493 0.81 DAO (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL24156586 0.78 PARP1 (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL24157206 0.78 TYMS (0.34) PDE3BPDE3ATYMSCASP3DAO
SCHEMBL30218641 0.78 PARP1 (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL25376579 0.75 TYMS (0.32) TYMSCASP3DAO
SCHEMBL31049737 0.75 TYMS (0.32) TYMSCASP3DAO
SCHEMBL14764904 0.74 CA12 (0.43) TYMSMAPTDAO
SCHEMBL24157258 0.73 KDM4E (0.36) NQO2PDE3BPDE3AGRIN2DGRIN3B
SCHEMBL30218627 0.73 KDM4E (0.36) NQO2PDE3BPDE3AGRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034758-A1 SUBSTITUTED TRIAZOLOPYRAZINES AND USES THEREOF H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed