SCHEMBL14768145

SCHEMBL14768145

CC(C)(O)c1cccc2c1ccn2-c1ccnc(NC2CCC(N)CC2)n1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 20/20 0.58
MAPK9 P45984 9/20 0.55
MAPK10 P53779 6/20 0.55
CCNE1 P24864 1/20 0.50
CDK2 P24941 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3807194 0.91 MAPK8 (0.66) MAPK8MAPK9MAPK10
SCHEMBL3807198 0.91 MAPK8 (0.66) MAPK8MAPK9MAPK10
SCHEMBL14768143 0.89 MAPK8 (0.59) MAPK8MAPK9MAPK10
SCHEMBL14768364 0.88 MAPK8 (0.66) MAPK8MAPK9MAPK10CCNE1CDK2
SCHEMBL5096255 0.88 MAPK8 (0.60) MAPK8MAPK9MAPK10
SCHEMBL14175777 0.88 MAPK8 (0.66) MAPK8MAPK9MAPK10CCNE1CDK2
SCHEMBL14175797 0.87 MAPK8 (0.69) MAPK8MAPK9MAPK10
SCHEMBL14768250 0.87 MAPK8 (0.69) MAPK8MAPK9MAPK10
SCHEMBL14175802 0.85 MAPK8 (0.67) MAPK8MAPK9MAPK10CCNE1CDK2
SCHEMBL14175793 0.84 MAPK8 (0.62) MAPK8MAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8399462-B2 4-[4-(4-benzyloxy-indol-1-yl)-pyrimidin-2-ylamino]-cyclohexanol; autoimmune, inflammatory, metabolic, neurological diseases as well as cancer and pain ROCHE PALO ALTO LLC (US) 2013-03-19 US disclosed