SCHEMBL14768389

SCHEMBL14768389

O=[SH](=O)NCc1ccc2cnn(-c3ccnc(NC4CCC(O)CC4)n3)c2c1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 17/20 0.66
MAPK9 P45984 15/20 0.66
MAPK10 P53779 13/20 0.66
CYP2C9 P11712 2/20 0.49
CCNE1 P24864 2/20 0.49
CDK2 P24941 2/20 0.49
MKNK1 Q9BUB5 3/20 0.46
MKNK2 Q9HBH9 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3814586 0.88 MAPK8 (0.70) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL5094240 0.88 MAPK8 (0.70) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL3805465 0.82 MAPK8 (0.73) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL5093840 0.82 MAPK8 (0.73) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL5090208 0.82 MAPK8 (0.73) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL3814615 0.82 MAPK8 (0.73) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL5102042 0.82 MAPK8 (0.69) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL14175785 0.80 MAPK8 (0.64) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL14768388 0.80 MAPK8 (0.64) MAPK8MAPK9MAPK10CYP2C9CCNE1
SCHEMBL5096150 0.80 MAPK8 (0.67) MAPK8MAPK9MAPK10CYP2C9CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8399462-B2 4-[4-(4-benzyloxy-indol-1-yl)-pyrimidin-2-ylamino]-cyclohexanol; autoimmune, inflammatory, metabolic, neurological diseases as well as cancer and pain ROCHE PALO ALTO LLC (US) 2013-03-19 US disclosed