Bicarbonate

Bicarbonate

SCHEMBL14775783

Cc1nn(C2CCOCC2)c2sc(C(=O)NC3CCCCC3)cc12.O=C(O)O

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 20/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL880652 0.98 PDE7A (0.85) PDE7A
Bicarbonate SCHEMBL14775793 0.93 PDE7A (0.84) PDE7A
Bicarbonate SCHEMBL14775802 0.93 PDE7A (0.84) PDE7A
SCHEMBL854148 0.91 PDE7A (0.88) PDE7A
SCHEMBL854150 0.91 PDE7A (0.88) PDE7A
SCHEMBL854018 0.91 PDE7A (1.00) PDE7A
SCHEMBL853402 0.89 PDE7A (0.82) PDE7A
SCHEMBL853401 0.89 PDE7A (0.82) PDE7A
SCHEMBL853480 0.89 PDE7A (0.78) PDE7A
SCHEMBL14776040 0.89 PDE7A (0.80) PDE7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1775298-B1 THIENOPYRAZOLE DERIVATIVE HAVING PDE7 INHIBITORY ACTIVITY DAIICHI SANKYO CO LTD (JP) 2013-03-20 EP claimed