SCHEMBL14780983

SCHEMBL14780983

Brc1ccc2nc(CI)ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.53
HDAC1 Q13547 5/20 0.47
HDAC2 Q92769 5/20 0.47
TLR2 O60603 1/20 0.40
CYP2A6 P11509 1/20 0.39
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
HTT P42858 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
PABPC1 P11940 1/20 0.35
PSMB5 P28074 1/20 0.35
NOS1 P29475 2/20 0.32
METAP2 P50579 2/20 0.32
CSNK2A1 P68400 1/20 0.32
DYRK1A Q13627 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27779108 0.85 BACE1 (0.53) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL2322461 0.82 BACE1 (0.55) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL14925243 0.81 BACE1 (0.53) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL30718905 0.81 BACE1 (0.53) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL1599323 0.81 BACE1 (0.53) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL5050008 0.81 BACE1 (0.53) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL1599686 0.81 BACE1 (0.58) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL27620530 0.79 BACE1 (0.52) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL14756191 0.78 BACE1 (0.55) BACE1HDAC1HDAC2TLR2CYP2A6
SCHEMBL1641368 0.78 BACE1 (0.50) BACE1HDAC1HDAC2TLR2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8399674-B2 Quinolines HOFFMAN-LA ROCHE INC. (US) 2013-03-19 US disclosed