SCHEMBL14796162

SCHEMBL14796162

Nc1c(-c2nc3cc(N4CCC[C@H]4CN4CCCC4)ccc3[nH]2)c(=O)[nH]c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 20/20 0.53
PDGFRB P09619 14/20 0.53
KDR P35968 14/20 0.53
FLT1 P17948 9/20 0.53
CHEK1 O14757 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14795575 0.84 FGFR1 (0.54) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL3384436 0.81 FGFR1 (0.70) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL3383616 0.78 FGFR1 (0.64) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL3383500 0.77 FGFR1 (0.64) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL3382790 0.77 FGFR1 (0.69) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL3384784 0.76 FGFR1 (0.87) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL3381227 0.76 FGFR1 (0.85) FGFR1PDGFRBKDRFLT1
SCHEMBL15910950 0.75 PDGFRB (0.48) FGFR1PDGFRBKDR
SCHEMBL3381125 0.75 FGFR1 (0.68) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL3383594 0.75 FGFR1 (0.55) FGFR1PDGFRBKDRFLT1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2762475-A1 Pharmaceutically acceptable salts of quinolinone compounds and their medical use Novartis Vaccines and Diagnostics, Inc. (US) 2014-08-06 EP disclosed
EP-2573079-A2 Benzimidazole quinolinones and uses thereof Novartis Vaccines and Diagnostics, Inc. (US) 2013-03-27 EP disclosed