SCHEMBL14796308

SCHEMBL14796308

COc1cc2[nH]c(-c3c(N)c4ccccc4[nH]c3=O)nc2cc1C

nearest known ligand 0.79

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 18/20 0.79
PDGFRB P09619 12/20 0.79
KDR P35968 12/20 0.79
FLT1 P17948 9/20 0.63
CHEK1 O14757 1/20 0.63
KDM4E B2RXH2 2/20 0.47
MAPT P10636 1/20 0.47
ATM Q13315 1/20 0.47
ALDH1A1 P00352 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4296125 0.89 FGFR1 (1.00) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL15911026 0.81 FGFR1 (0.67) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL1054595 0.81 FGFR1 (1.00) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL4291574 0.79 FGFR1 (0.74) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL1050162 0.78 FGFR1 (1.00) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL30737932 0.78 FGFR1 (1.00) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL1054179 0.78 FGFR1 (0.68) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL13041327 0.77 FGFR1 (0.68) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL1055032 0.76 FGFR1 (0.74) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL4287779 0.76 FGFR1 (0.65) FGFR1PDGFRBKDRFLT1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2762475-A1 Pharmaceutically acceptable salts of quinolinone compounds and their medical use Novartis Vaccines and Diagnostics, Inc. (US) 2014-08-06 EP disclosed
EP-2573079-A2 Benzimidazole quinolinones and uses thereof Novartis Vaccines and Diagnostics, Inc. (US) 2013-03-27 EP disclosed