Bicarbonate

Bicarbonate

SCHEMBL14796763

Fc1cc2nc(-c3ccc(Cl)cc3)n(C(COc3ccc(OC4CC4)cn3)C3CCCCC3)c2cc1F.O=C(O)O

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.53
CYP2C9 P11712 7/20 0.53
CYP3A4 P08684 5/20 0.53
CYP2D6 P10635 5/20 0.53
KCNH2 Q12809 5/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL14796784 0.92 NR1H4 (0.56) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL197863 0.90 NR1H4 (0.53) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
Bicarbonate SCHEMBL14796775 0.89 NR1H4 (0.55) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL197563 0.88 NR1H4 (0.65) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL199161 0.88 NR1H4 (0.65) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL14796894 0.88 NR1H4 (0.54) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL197524 0.88 NR1H4 (0.51) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL197219 0.88 NR1H4 (0.51) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL197666 0.88 NR1H4 (0.64) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL14796796 0.86 NR1H4 (0.49) NR1H4CYP2C9CYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-B1 NEW BENZIMIDAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2013-03-27 EP claimed