SCHEMBL14797019

SCHEMBL14797019

Cc1cc(-c2nc3cnc(Oc4ccccc4F)nc3o2)ccc1OCC(=O)O

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.56
PPARD Q03181 8/20 0.44
FFAR1 O14842 1/20 0.44
PPARA Q07869 5/20 0.43
PPARG P37231 4/20 0.43
MAPT P10636 3/20 0.43
RXFP1 Q9HBX9 2/20 0.43
LMNA P02545 1/20 0.43
S1PR5 Q9H228 1/20 0.43
CEPT1 Q9Y6K0 4/20 0.43
TP53 P04637 2/20 0.43
THRB P10828 1/20 0.43
HPGD P15428 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CETP P11597 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2225216 0.90 S1PR1 (0.69) S1PR1PPARDFFAR1PPARAPPARG
SCHEMBL2223582 0.88 S1PR1 (0.47) S1PR1PPARDFFAR1PPARAPPARG
SCHEMBL2226787 0.86 S1PR1 (0.51) S1PR1PPARDFFAR1PPARAPPARG
SCHEMBL2228824 0.86 S1PR1 (0.42) S1PR1MAPTRXFP1LMNAS1PR5
SCHEMBL14797105 0.85 S1PR1 (0.65) S1PR1PPARDFFAR1CEPT1CETP
SCHEMBL14777954 0.84 KMT2A (0.44) S1PR1MAPTRXFP1LMNAS1PR5
SCHEMBL2223287 0.84 KMT2A (0.44) S1PR1MAPTRXFP1LMNAS1PR5
SCHEMBL2223289 0.84 S1PR1 (0.42) S1PR1MAPTRXFP1LMNAS1PR5
SCHEMBL2225375 0.84 S1PR1 (0.44) S1PR1MAPTRXFP1LMNACEPT1
SCHEMBL14797018 0.83 S1PR1 (0.65) S1PR1PPARDFFAR1PPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8846692-B2 Carboxylic acid derivatives having a 2,5-substituted oxazolopyrimidine ring SANOFI (FR) 2014-09-30 US disclosed
US-20130079358-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI (FR) 2013-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130079358-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING OXGR1, EDNRA, EDF1 S1PR1 129/4885PPARD 370/4885FFAR1 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.