SCHEMBL1484253

SCHEMBL1484253

COC1=CC(c2cccc(OC)c2)=CCC1(N=C=O)N=C=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
HDAC4 P56524 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
DYRK1A Q13627 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
GAA P10253 3/20 0.35
ALDH1A1 P00352 3/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
GSK3B P49841 1/20 0.34
GALR1 P47211 1/20 0.33
NISCH Q9Y2I1 1/20 0.33
PGR P06401 1/20 0.33
ERN1 O75460 1/20 0.33
BRD4 O60885 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL912114 0.66 HDAC4 (0.35) NCOA1NCOA3HDAC4HDAC8DYRK1A
SCHEMBL14993 0.64 HDAC4 (0.58) HDAC4HDAC8DYRK1ACLK4GAA
SCHEMBL9869408 0.64 HDAC4 (0.58) HDAC4HDAC8DYRK1ACLK4GAA
SCHEMBL30185444 0.64 HDAC4 (0.58) HDAC4HDAC8DYRK1ACLK4GAA
SCHEMBL26486027 0.64 DYRK1A (0.42) NCOA1NCOA3HDAC4HDAC8DYRK1A
SCHEMBL196765 0.63 CYP3A4 (0.73) HDAC4HDAC8DYRK1ACLK4GAA
SCHEMBL29489425 0.63 CYP3A4 (0.73) HDAC4HDAC8DYRK1ACLK4GAA
SCHEMBL5887546 0.62 DYRK1A (0.44) NCOA1NCOA3HDAC4HDAC8DYRK1A
SCHEMBL29628977 0.61 CYP3A4 (0.77) HDAC4HDAC8DYRK1ACLK4GAA
Ammonia Solution, Strong SCHEMBL27960505 0.61 CYP3A4 (0.70) HDAC4HDAC8DYRK1ACLK4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024033289-A1 A PHOTOCURABLE OLIGOMER CONTAINING URETDIONE GROUPS, METHOD OF PREPARING THE OLIGOMER AND DUAL-CURE RESIN COMPOSITION CONTAINING THE OLIGOMER THEREOF BASF SE (DE) 2024-02-15 WO claimed
US-8394567-B2 Toner, developer, toner cartridge, process cartridge, and image forming apparatus FUJI XEROX CO., LTD. (JP) 2013-03-12 US claimed
EP-4739723-A1 MULTI-COMPONENT RESIN SYSTEM COMPRISING AT LEAST ONE MONOALCOHOL, MORTAR COMPOSITION BASED ON ISOCYANATE-AMINE ADDUCTS, AND METHOD AND USE OF THE MULTI-COMPONENT RESIN SYSTEM FOR FASTENING CONSTRUCTION ELEMENTS Hilti Aktiengesellschaft (LI) 2026-05-13 EP disclosed
WO-2025008202-A1 MULTI-COMPONENT RESIN SYSTEM COMPRISING AT LEAST ONE MONOALCOHOL, MORTAR COMPOSITION BASED ON ISOCYANATE-AMINE ADDUCTS, AND METHOD AND USE OF THE MULTI-COMPONENT RESIN SYSTEM FOR FASTENING CONSTRUCTION ELEMENTS HILTI AKTIENGESELLSCHAFT (LI) 2025-01-09 WO disclosed
CN-117321110-A Polyurethane foam and cushioning material 井上株式会社 2023-12-29 CN disclosed
CN-116368200-A Polyurethane foam and toner sealing member 井上株式会社 2023-06-30 CN disclosed
CN-112154166-B Polyurethane-polyisocyanurate foam 陶氏环球技术有限责任公司 2023-04-04 CN disclosed
CN-112638980-B Method for reducing aldehyde emissions in polyurethane foams 陶氏环球技术有限责任公司 2023-03-31 CN disclosed
CN-113272363-B Silicone-organic copolymers, sealants including silicone-organic copolymers, and related methods 美国陶氏有机硅公司 2023-02-17 CN disclosed
US-20230048616-A1 INK COMPOSITION FOR WATER-BASED BALLPOINT PENS MITSUBISHI PENCIL COMPANY, LIMITED (JP) 2023-02-16 US disclosed
CN-112166140-B Process for preparing alkoxylation products 巴克莱特有限公司 2023-02-07 CN disclosed
US-5070110-A REACTION INJECTION MOLDED POLYURETHANES HAVING SHORT DEMOLD TI MES THE DOW CHEMICAL COMPANY (US) 1991-12-03 US disclosed
EP-0152699-B1 AN ANTITHROMBOGENIC POLYURETHANE POLYMER AND A PROCESS FOR IMPARTING ANTITHROMBOGENIC ACTIVITY TO A POLYURETHANE SUBSTRATE Deseret Medical, Inc. (US) 1990-06-06 EP disclosed
US-4720512-A AMINE, HYDROPHOBIC, PLASMA BECTON, DICKINSON AND COMPANY (US) 1988-01-19 US disclosed
US-4713402-A USING DUAL SOLVENT SYSTEM OF CHLOROFLUOROCARBON AND PETROLEUM ETHER BECTON, DICKINSON AND COMPANY (US) 1987-12-15 US disclosed
US-4678660-A MEDICAL EQUIPMENT DESERET MEDICAL, INC. (US) 1987-07-07 US disclosed
US-4676975-A Thermoplastic polyurethane anticoagulant alloy coating BECTON, DICKINSON AND COMPANY (US) 1987-06-30 US disclosed
US-4600652-A Permanently bonded antithrombogenic polyurethane surface WARNER-LAMBERT COMPANY (US) 1986-07-15 US disclosed
EP-0184465-A2 A thermoplastic polyurethane product Deseret Medical, Inc. (US) 1986-06-11 EP disclosed
US-4521564-A BONDING POLYURETHANE TO POLYMERIC AMINE, THEN BONING ANTICOAGULANT WARNER-LAMBERT COMPANY (US) 1985-06-04 US disclosed