SCHEMBL14844178

SCHEMBL14844178

COc1ccc2ncc(N3CC4CC(CN(C(=O)c5cc(C)ccc5-n5nccn5)C4)C3)nc2c1

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 20/20 0.65
HCRTR1 O43613 19/20 0.65
KCNH2 Q12809 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14844230 0.97 HCRTR2 (0.65) HCRTR2HCRTR1KCNH2
SCHEMBL14844170 0.88 HCRTR2 (0.57) HCRTR2HCRTR1
SCHEMBL14844332 0.88 HCRTR1 (0.61) HCRTR2HCRTR1
SCHEMBL14844206 0.88 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL14844268 0.85 HCRTR2 (0.57) HCRTR2HCRTR1
SCHEMBL14844341 0.85 HCRTR1 (0.61) HCRTR2HCRTR1
SCHEMBL14844159 0.82 HCRTR2 (0.57) HCRTR2HCRTR1
SCHEMBL1671957 0.79 HCRTR1 (1.00) HCRTR2HCRTR1KCNH2
SCHEMBL14843945 0.77 HCRTR2 (0.66) HCRTR2HCRTR1
SCHEMBL4312445 0.77 HCRTR2 (0.75) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013050938-A1 3,7-DIAZABICYCLO[3.3.1]NONANE AND 9-OXA-3,7-DIAZABICYCLO[3.3.1]NONANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2013-04-11 WO claimed
WO-2013050938-A1 3,7-DIAZABICYCLO[3.3.1]NONANE AND 9-OXA-3,7-DIAZABICYCLO[3.3.1]NONANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2013-04-11 WO disclosed