SCHEMBL14856751

SCHEMBL14856751

CC(C)c1cc(C(=O)N2CCC(N)CC2)c(O)cc1O

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.67
HSP90AB1 P08238 7/20 0.67
HSP90B1 P14625 5/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15000795 0.87 HSP90AA1 (0.68) HSP90AA1HSP90AB1HSP90B1
SCHEMBL488032 0.84 HSP90AA1 (0.64) HSP90AA1HSP90AB1HSP90B1
SCHEMBL14856614 0.83 HSP90AA1 (0.60) HSP90AA1HSP90AB1HSP90B1
SCHEMBL487633 0.82 HSP90AA1 (0.61) HSP90AA1HSP90AB1HSP90B1
SCHEMBL10256085 0.82 HSP90AA1 (0.61) HSP90AA1HSP90AB1HSP90B1
SCHEMBL10256000 0.82 HSP90AA1 (0.61) HSP90AA1HSP90AB1HSP90B1
SCHEMBL10256936 0.82 HSP90AA1 (0.61) HSP90AA1HSP90AB1HSP90B1
SCHEMBL487588 0.81 HSP90AA1 (0.72) HSP90AA1HSP90AB1HSP90B1
SCHEMBL487620 0.81 HSP90AA1 (0.72) HSP90AA1HSP90AB1HSP90B1
SCHEMBL14856436 0.81 HSP90AA1 (0.60) HSP90AA1HSP90AB1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2580193-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS HSP90 INHIBTORS Chroma Therapeutics Ltd. (GB) 2013-04-17 EP disclosed
WO-2011154708-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS HSP90 INHIBTORS CHROMA THERAPEUTICS LTD (GB) 2011-12-15 WO disclosed