SCHEMBL14865316

SCHEMBL14865316

CC=C(NCc1ncc(Nc2ccc(Cl)cc2C(F)(F)F)cc1F)[C@]1(NC(=O)c2cnc(NC)nc2)CCOC1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 8/20 0.34
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
TP53 P04637 2/20 0.32
LRRK2 Q5S007 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
HDAC3 O15379 2/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC2 Q92769 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
GNRHR P30968 1/20 0.31
PTK2 Q05397 2/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
P2RX3 P56373 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2812255 0.93 CNR2 (0.35) CNR2CYP1A2CYP3A4CYP2C9TP53
SCHEMBL2805186 0.86 CNR2 (0.37) CNR2CYP1A2CYP3A4CYP2C9TP53
SCHEMBL2810858 0.86 CNR2 (0.38) CNR2CYP1A2CYP3A4CYP2C9TP53
SCHEMBL2807388 0.84 BDKRB1 (0.39) CNR2CYP1A2TP53CYP2D6CYP2C19
SCHEMBL2809124 0.83 CNR2 (0.36) CNR2CYP1A2CYP3A4CYP2C9TP53
SCHEMBL186328 0.83 CNR2 (0.35) CNR2CYP1A2CYP3A4CYP2C9TP53
SCHEMBL2805102 0.83 CNR2 (0.35) CNR2CYP1A2CYP3A4CYP2C9TP53
SCHEMBL13129178 0.83 CNR2 (0.37) CNR2CYP1A2TP53CYP2D6CYP2C19
SCHEMBL2806938 0.82 HDAC3 (0.37) CNR2LRRK2HDAC3HDAC1HDAC2
SCHEMBL2805933 0.82 PTK2 (0.42) CNR2CYP1A2CYP3A4CYP2C9LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed