SCHEMBL14865367

SCHEMBL14865367

Cc1ncc(C(=O)N[C@@]2(C(=O)NCc3ncc(Nc4ccc(F)cc4C(F)(F)I)cc3C)CCOC2)cn1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.34
HDAC3 O15379 4/20 0.32
HDAC1 Q13547 4/20 0.32
HDAC2 Q92769 4/20 0.32
HDAC6 Q9UBN7 4/20 0.32
RAF1 P04049 7/20 0.30
BRAF P15056 1/20 0.30
PDE2A O00408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2808146 0.94 OPRL1 (0.38) OPRL1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2805565 0.88 OPRL1 (0.38) OPRL1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2805695 0.88 OPRL1 (0.37) OPRL1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2807541 0.87 DHODH (0.35) OPRL1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2810028 0.87 CNR2 (0.40) PDE2A
SCHEMBL2805193 0.86 HDAC3 (0.38) OPRL1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2809544 0.84 OPRL1 (0.39) OPRL1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2809999 0.84 BDKRB1 (0.36) OPRL1RAF1BRAFPDE2A
SCHEMBL185964 0.84 BDKRB1 (0.36) OPRL1RAF1BRAFPDE2A
SCHEMBL185516 0.83 OPRL1 (0.36) OPRL1RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed