SCHEMBL14878664

SCHEMBL14878664

CNc1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.79
ERBB2 P04626 15/20 0.79
GAK O14976 1/20 0.76
ERBB4 Q15303 2/20 0.72
ERBB3 P21860 1/20 0.66
ABL1 P00519 2/20 0.64
INSR P06213 2/20 0.64
PDGFRB P09619 2/20 0.64
CDK2 P24941 2/20 0.64
PLK1 P53350 2/20 0.64
HDAC1 Q13547 2/20 0.64
HDAC8 Q9BY41 2/20 0.64
HDAC6 Q9UBN7 2/20 0.64
HDAC3 O15379 1/20 0.64
HDAC4 P56524 1/20 0.64
HDAC7 Q8WUI4 1/20 0.64
HDAC2 Q92769 1/20 0.64
HDAC10 Q969S8 1/20 0.64
HDAC11 Q96DB2 1/20 0.64
HDAC9 Q9UKV0 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12691367 0.90 EGFR (0.76) EGFRERBB2GAKERBB4ERBB3
SCHEMBL24535497 0.90 EGFR (0.75) EGFRERBB2GAKERBB4ERBB3
SCHEMBL2510931 0.89 EGFR (0.75) EGFRERBB2GAKERBB4ERBB3
SCHEMBL2505296 0.89 EGFR (0.77) EGFRERBB2GAKERBB4ERBB3
SCHEMBL14509726 0.89 EGFR (0.75) EGFRERBB2GAKERBB4ERBB3
SCHEMBL233913 0.89 EGFR (0.77) EGFRERBB2GAKERBB4ERBB3
SCHEMBL6954367 0.89 EGFR (0.80) EGFRERBB2GAKERBB4ERBB3
SCHEMBL9973598 0.89 EGFR (0.73) EGFRERBB2GAKERBB4ERBB3
SCHEMBL141514 0.89 EGFR (0.73) EGFRERBB2GAKERBB4ERBB3
SCHEMBL29693649 0.89 EGFR (0.73) EGFRERBB2GAKERBB4ERBB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2248806-B1 Quinazoline derivatives as tyrosine kinase inhibitors SHANGHAI ALLIST PHARMACEUTICALS INC (CN) 2013-04-24 EP disclosed