SCHEMBL1488958

SCHEMBL1488958

CCN(C(=O)c1cccc(Cl)c1F)c1nnc(-c2cc(C)c(OCCN3CCC(C(=O)O)CC3)c(C)c2)s1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.50
S1PR3 Q99500 6/20 0.50
S1PR4 O95977 1/20 0.43
S1PR5 Q9H228 1/20 0.43
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1489155 0.99 S1PR1 (0.49) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1489168 0.93 S1PR1 (0.60) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1488835 0.93 S1PR1 (0.57) S1PR1S1PR3S1PR4S1PR5KDM4E
Hydrochloric Acid SCHEMBL1489221 0.92 S1PR1 (0.57) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1489136 0.91 S1PR1 (0.60) S1PR1S1PR3S1PR4S1PR5
Hydrochloric Acid SCHEMBL1647422 0.90 S1PR1 (0.59) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1488857 0.87 S1PR1 (0.62) S1PR1S1PR3S1PR4S1PR5ALDH1A1
SCHEMBL1488910 0.87 S1PR1 (0.54) S1PR1S1PR3S1PR4S1PR5ALDH1A1
SCHEMBL1488863 0.87 S1PR1 (0.54) S1PR1S1PR3S1PR4S1PR5ALDH1A1
Hydrochloric Acid SCHEMBL1647928 0.86 S1PR1 (0.54) S1PR1S1PR3S1PR4S1PR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2305660-A1 New thiadiazole derivatives Almirall, S.A. (ES) 2011-04-06 EP claimed
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO claimed
EP-2305660-A1 New thiadiazole derivatives Almirall, S.A. (ES) 2011-04-06 EP disclosed
EP-2305660-A1 New thiadiazole derivatives Almirall, S.A. (ES) 2011-04-06 EP disclosed
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO disclosed
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO disclosed