SCHEMBL1489208

SCHEMBL1489208

CCCCN(C(=O)Cc1ccccc1OC)c1nnc(-c2ccc(CN3CC(C(=O)O)C3)cc2)s1

nearest known ligand 0.80

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.80
S1PR3 Q99500 6/20 0.69
S1PR4 O95977 1/20 0.68
S1PR5 Q9H228 1/20 0.68
CPB1 P15086 1/20 0.63
KDM4E B2RXH2 2/20 0.56
MEN1 O00255 1/20 0.56
CYP1A2 P05177 1/20 0.56
GAA P10253 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
KMT2A Q03164 1/20 0.56
USP2 O75604 1/20 0.46
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1647943 0.90 S1PR1 (0.70) S1PR1S1PR3S1PR4S1PR5CPB1
SCHEMBL1966067 0.89 S1PR1 (1.00) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1966214 0.89 S1PR1 (0.81) S1PR1S1PR3S1PR4S1PR5CPB1
SCHEMBL1964964 0.89 S1PR1 (1.00) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1965766 0.84 S1PR1 (1.00) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1964578 0.83 S1PR1 (0.78) S1PR1S1PR3S1PR4S1PR5CPB1
SCHEMBL1488768 0.82 S1PR1 (0.60) S1PR1S1PR3S1PR4S1PR5CPB1
SCHEMBL1966144 0.82 S1PR1 (0.85) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1965502 0.82 S1PR1 (1.00) S1PR1S1PR3S1PR4S1PR5
Hydrochloric Acid SCHEMBL1488907 0.82 S1PR1 (0.59) S1PR1S1PR3S1PR4S1PR5CPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2305660-A1 New thiadiazole derivatives Almirall, S.A. (ES) 2011-04-06 EP claimed
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO claimed
EP-2305660-A1 New thiadiazole derivatives Almirall, S.A. (ES) 2011-04-06 EP disclosed
EP-2305660-A1 New thiadiazole derivatives Almirall, S.A. (ES) 2011-04-06 EP disclosed
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO disclosed
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO disclosed