SCHEMBL1489689

SCHEMBL1489689

NC(=O)OC1CCCN(CC(=O)Nc2cc(-c3nccs3)nc(-c3cccs3)n2)C1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.51
ADORA1 P30542 16/20 0.51
ADORA3 P0DMS8 3/20 0.44
HPGD P15428 1/20 0.41
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490245 0.91 ADORA2A (0.56) ADORA2AADORA1ADORA3HPGDCYP3A4
SCHEMBL1489988 0.89 ADORA2A (0.53) ADORA2AADORA1CYP3A4
SCHEMBL1489712 0.88 ADORA2A (0.53) ADORA2AADORA1ADORA3HPGDCYP3A4
SCHEMBL1489658 0.86 ADORA2A (0.57) ADORA2AADORA1ADORA3HPGDCYP3A4
SCHEMBL1490173 0.86 ADORA2A (0.70) ADORA2AADORA1
SCHEMBL1489218 0.85 ADORA2A (0.65) ADORA2AADORA1ADORA3HPGDCYP3A4
SCHEMBL1489853 0.84 ADORA2A (0.53) ADORA2AADORA1ADORA3HPGDCYP3A4
SCHEMBL1489159 0.84 ADORA2A (0.64) ADORA2AADORA1ADORA3HPGDCYP3A4
SCHEMBL1489383 0.84 ADORA2A (0.64) ADORA2AADORA1ADORA3HPGDCYP3A4
SCHEMBL1489812 0.83 ADORA2A (0.59) ADORA2AADORA1ADORA3HPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888565-B1 2, 6-DI (HETERO) ARYL -4-AMIDO-PYRIMIDINES AS ADENOSINE RECEPTOR ANTAGONISTS ALMIRALL SA (ES) 2011-03-23 EP claimed