SCHEMBL1489937

SCHEMBL1489937

Cc1ccc(-c2nc(NC(=O)CN3CCC(OC(N)=O)CC3)cc(-c3nccs3)n2)o1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 19/20 0.75
ADORA2A P29274 19/20 0.75
KCNH2 Q12809 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490173 0.92 ADORA2A (0.70) ADORA1ADORA2AKCNH2
SCHEMBL1489193 0.91 ADORA2A (0.79) ADORA1ADORA2AKCNH2
SCHEMBL1489062 0.90 ADORA2A (0.82) ADORA1ADORA2AKCNH2
SCHEMBL1489710 0.90 ADORA2A (0.79) ADORA1ADORA2AKCNH2
SCHEMBL1490175 0.89 ADORA1 (0.70) ADORA1ADORA2AKCNH2
SCHEMBL1489496 0.89 ADORA2A (0.82) ADORA1ADORA2AKCNH2
SCHEMBL1489289 0.89 ADORA2A (0.82) ADORA1ADORA2AKCNH2
SCHEMBL1489705 0.88 ADORA2A (0.79) ADORA1ADORA2AKCNH2
SCHEMBL1490030 0.88 ADORA2A (0.90) ADORA1ADORA2AKCNH2
SCHEMBL1489645 0.87 ADORA2A (0.88) ADORA1ADORA2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888565-B1 2, 6-DI (HETERO) ARYL -4-AMIDO-PYRIMIDINES AS ADENOSINE RECEPTOR ANTAGONISTS ALMIRALL SA (ES) 2011-03-23 EP claimed