SCHEMBL1490101

SCHEMBL1490101

Cc1cc(C)n(-c2cc(NC(=O)CN3CC[C@H](N(C)C)C3)nc(-c3occc3C)n2)n1

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.74
ADORA1 P30542 20/20 0.74
KCNH2 Q12809 7/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1489872 0.85 ADORA2A (1.00) ADORA2AADORA1KCNH2
SCHEMBL1489628 0.85 ADORA2A (1.00) ADORA2AADORA1KCNH2
SCHEMBL1489626 0.85 ADORA2A (1.00) ADORA2AADORA1KCNH2
SCHEMBL1489926 0.83 ADORA2A (0.73) ADORA2AADORA1KCNH2
SCHEMBL1489924 0.83 ADORA2A (0.73) ADORA2AADORA1KCNH2
SCHEMBL1490032 0.83 ADORA2A (0.73) ADORA2AADORA1KCNH2
SCHEMBL1489299 0.81 ADORA2A (0.92) ADORA2AADORA1KCNH2
SCHEMBL1489295 0.81 ADORA2A (0.92) ADORA2AADORA1KCNH2
SCHEMBL1489779 0.81 ADORA2A (0.74) ADORA2AADORA1KCNH2
SCHEMBL1489782 0.81 ADORA2A (0.92) ADORA2AADORA1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888565-B1 2, 6-DI (HETERO) ARYL -4-AMIDO-PYRIMIDINES AS ADENOSINE RECEPTOR ANTAGONISTS ALMIRALL SA (ES) 2011-03-23 EP claimed