SCHEMBL1490125

SCHEMBL1490125

Cc1ccc(-c2nc(NC(=O)CN3CCN(CC(=O)C(C)C)CC3)cc(-c3ccccn3)n2)o1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.61
ADORA1 P30542 19/20 0.61
KCNH2 Q12809 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1489532 0.91 ADORA2A (0.61) ADORA2AADORA1KCNH2
SCHEMBL1489303 0.90 ADORA2A (0.73) ADORA2AADORA1KCNH2
SCHEMBL1489765 0.90 ADORA2A (0.63) ADORA2AADORA1KCNH2
SCHEMBL1489538 0.89 ADORA2A (0.63) ADORA2AADORA1KCNH2
SCHEMBL1489531 0.87 ADORA2A (0.56) ADORA2AADORA1KCNH2
SCHEMBL1489731 0.85 ADORA2A (0.57) ADORA2AADORA1KCNH2
SCHEMBL1489343 0.84 ADORA2A (0.57) ADORA2AADORA1KCNH2
SCHEMBL1489438 0.83 ADORA2A (0.55) ADORA2AADORA1KCNH2
SCHEMBL1489768 0.83 ADORA2A (0.55) ADORA2AADORA1KCNH2
SCHEMBL4962442 0.80 ADORA2A (0.55) ADORA2AADORA1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888565-B1 2, 6-DI (HETERO) ARYL -4-AMIDO-PYRIMIDINES AS ADENOSINE RECEPTOR ANTAGONISTS ALMIRALL SA (ES) 2011-03-23 EP claimed