SCHEMBL14901457

SCHEMBL14901457

COc1cc(OC)c(F)c(N(CC(O)CO)c2ccc3ncc(-c4cnn(CC(O)COC(C)C)c4)nc3n2)c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 20/20 0.51
FGFR2 P21802 20/20 0.51
FGFR4 P22455 20/20 0.51
FGFR3 P22607 20/20 0.51
KDR P35968 17/20 0.51
VEGFA P15692 3/20 0.43
FLT1 P17948 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16125196 0.97 FGFR1 (0.52) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL14901360 0.88 FGFR1 (0.61) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL14901261 0.88 FGFR1 (0.61) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL14901246 0.87 FGFR1 (0.59) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL16125195 0.84 FGFR3 (0.56) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL16125129 0.83 FGFR1 (0.45) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL20309577 0.82 FGFR1 (0.62) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL20306121 0.82 FGFR1 (0.44) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL20309779 0.82 FGFR3 (0.54) FGFR1FGFR2FGFR4FGFR3KDR
SCHEMBL14901321 0.82 FGFR1 (0.60) FGFR1FGFR2FGFR4FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013061080-A1 ANTICANCER PYRIDOPYRAZINES VIA THE INHIBITION OF FGFR KINASES ASTEX THERAPEUTICS LIMITED (GB) 2013-05-02 WO disclosed