SCHEMBL1490436

SCHEMBL1490436

Cc1ccc(-c2scc(NC(=O)c3ccc(Cl)cc3)c2C(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
LMNA P02545 2/20 0.52
POLB P06746 2/20 0.52
KMT2A Q03164 10/20 0.49
MEN1 O00255 9/20 0.49
RAB9A P51151 7/20 0.49
NPC1 O15118 7/20 0.49
GRIN2C Q14957 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
ALDH1A1 P00352 3/20 0.47
HPGD P15428 2/20 0.47
HTT P42858 2/20 0.47
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
ANO1 Q5XXA6 2/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490465 1.00 MAPT (0.52) MAPTLMNAPOLBKMT2AMEN1
SCHEMBL1490509 0.94 KMT2A (0.55) MAPTLMNAKMT2AMEN1RAB9A
SCHEMBL1490816 0.94 MAPT (0.58) MAPTLMNAPOLBKMT2AMEN1
SCHEMBL12756545 0.89 ANO1 (0.49) MAPTLMNAKMT2AMEN1RAB9A
SCHEMBL1490373 0.89 KMT2A (0.52) MAPTLMNAKMT2AMEN1RAB9A
SCHEMBL12756874 0.88 NPC1 (0.64) MAPTLMNAPOLBKMT2AMEN1
SCHEMBL1490583 0.88 MEN1 (0.49) MAPTLMNAKMT2AMEN1RAB9A
SCHEMBL1490525 0.88 MEN1 (0.64) MAPTLMNAPOLBKMT2AMEN1
SCHEMBL1490520 0.88 MEN1 (0.49) MAPTLMNAKMT2AMEN1RAB9A
SCHEMBL1490609 0.88 NPC1 (0.64) MAPTLMNAPOLBKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140051711-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2014-02-20 US disclosed
US-8618307-B2 Compounds that modulate intracellular calcium CALCIMEDICA, INC. (US) 2013-12-31 US disclosed
EP-2477982-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2012-07-25 EP disclosed
WO-2011034962-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2011-03-24 WO disclosed
US-20110065724-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2011-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140051711-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM ORAI1, SARAF, RYR2 MAPT 1478/4885LMNA 1306/4885POLB 4774/4885
US-20110065724-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM ORAI1, SARAF, RYR2 MAPT 1478/4885LMNA 1306/4885POLB 4774/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.