SCHEMBL14905693

SCHEMBL14905693

Cc1c(C(Nc2ccc(C(=O)O)cc2)C2CCCCC2)sc2cnccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RCE1 Q9Y256 2/20 0.45
CSNK2A1 P68400 3/20 0.40
CSNK2A2 P19784 2/20 0.40
CSNK2B P67870 2/20 0.40
PDE7A Q13946 1/20 0.38
LCK P06239 1/20 0.38
JAK3 P52333 1/20 0.38
MERTK Q12866 1/20 0.36
NAMPT P43490 1/20 0.35
HIPK2 Q9H2X6 2/20 0.35
AKT1 P31749 1/20 0.35
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
FPR2 P25090 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
LTA4H P09960 1/20 0.33
POLB P06746 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14905709 0.92 RCE1 (0.45) RCE1CSNK2A1CSNK2A2CSNK2BPDE7A
SCHEMBL717365 0.87 GCG (0.48)
SCHEMBL716694 0.86 NAMPT (0.35) RCE1PDE7ALCKJAK3NAMPT
SCHEMBL720764 0.86 RCE1 (0.46) RCE1PDE7AMERTKPOLBKDM4E
SCHEMBL718249 0.85 RCE1 (0.44) RCE1PDE7AMERTKKDM4E
SCHEMBL720081 0.82 MEN1 (0.41) PDE7A
SCHEMBL719154 0.81 GCG (0.43)
SCHEMBL719453 0.81 RCE1 (0.60) RCE1PDE7ALCKJAK3MERTK
SCHEMBL718563 0.81 NAMPT (0.34) RCE1PDE7ALCKJAK3NAMPT
SCHEMBL14905663 0.80 RCE1 (0.54) RCE1PDE7ALCKJAK3MERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8436043-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-05-07 US disclosed