SCHEMBL14909545

SCHEMBL14909545

CCCC[C@H](CN(C(=O)O)C(C)(C)C)Nc1nc(Cl)c(C#N)cc1F

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KHK P50053 1/20 0.33
KCNH2 Q12809 3/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
POLB P06746 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14909546 1.00 KHK (0.33) KHKKCNH2L3MBTL1POLBKDM4E
SCHEMBL14908691 0.94 KHK (0.34) KHKKCNH2
SCHEMBL14908690 0.94 KHK (0.34) KHKKCNH2
SCHEMBL14909162 0.90 KHK (0.34) KHK
SCHEMBL14909161 0.90 KHK (0.34) KHK
SCHEMBL14911504 0.87 KHK (0.34) KHK
SCHEMBL14909516 0.87 KHK (0.34) KHK
SCHEMBL14908685 0.87 KHK (0.34) KHK
SCHEMBL14910363 0.84 KHK (0.37) KHK
SCHEMBL14910361 0.84 KHK (0.37) KHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2589592-B1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM CORP (JP) 2018-08-22 EP disclosed
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-8772320-B2 2014-07-08 US disclosed
EP-2589592-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM Corporation (JP) 2013-05-08 EP disclosed