SCHEMBL14918147

SCHEMBL14918147

Cc1nn(-c2ccc(C(N)=O)c(NCC3CCNCC3)c2)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 15/20 0.66
HSP90AB1 P08238 15/20 0.66
HSP90B1 P14625 4/20 0.56
TRAP1 Q12931 4/20 0.56
OPRM1 P35372 4/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1220533 0.94 HSP90AB1 (0.71) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1
SCHEMBL14918499 0.89 HSP90AB1 (0.64) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1
SCHEMBL16883488 0.85 HSP90AB1 (0.73) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1
SCHEMBL14932861 0.85 HSP90AB1 (0.59) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1
SCHEMBL1219235 0.85 HSP90AB1 (0.61) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1
SCHEMBL16161829 0.84 HSP90AB1 (0.77) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1
SCHEMBL1220688 0.84 HSP90AB1 (0.77) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL1220613 0.84 HSP90AA1 (0.68) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1
SCHEMBL1219504 0.84 HSP90AA1 (0.68) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1
SCHEMBL1220784 0.84 HSP90AA1 (0.68) HSP90AA1HSP90AB1HSP90B1TRAP1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013066831-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2013-05-10 WO disclosed
WO-2013066831-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2013-05-10 WO disclosed