SCHEMBL14920501

SCHEMBL14920501

Cc1nc(N)nc2c1C(=NO)C[C@@H](c1ccc(F)cc1-c1cccnc1)C2

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.44
HSP90AB1 P08238 8/20 0.42
TRAP1 Q12931 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12075133 1.00 HSP90AA1 (0.44) HSP90AA1HSP90AB1TRAP1
SCHEMBL14920498 1.00 HSP90AA1 (0.44) HSP90AA1HSP90AB1TRAP1
SCHEMBL1781588 1.00 HSP90AA1 (0.44) HSP90AA1HSP90AB1TRAP1
SCHEMBL1781589 1.00 HSP90AA1 (0.44) HSP90AA1HSP90AB1TRAP1
SCHEMBL14921019 1.00 HSP90AA1 (0.44) HSP90AA1HSP90AB1TRAP1
SCHEMBL14921203 1.00 HSP90AA1 (0.44) HSP90AA1HSP90AB1TRAP1
SCHEMBL14921201 1.00 HSP90AA1 (0.44) HSP90AA1HSP90AB1TRAP1
SCHEMBL1780042 0.91 HSP90AA1 (0.47) HSP90AA1HSP90AB1TRAP1
SCHEMBL1780040 0.91 HSP90AA1 (0.47) HSP90AA1HSP90AB1TRAP1
SCHEMBL1782639 0.90 HSP90AA1 (0.41) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013064919-A1 QUINAZOLINE DERIVATIVES WITH HSP90 INHIBITORY ACTIVITY DAC SRL (IT) 2013-05-10 WO claimed
WO-2013064919-A1 QUINAZOLINE DERIVATIVES WITH HSP90 INHIBITORY ACTIVITY DAC SRL (IT) 2013-05-10 WO disclosed