SCHEMBL14923699

SCHEMBL14923699

C[C@H](N)[C@@H](C)NC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA7 P43166 2/20 0.50
CYP2D6 P10635 1/20 0.45
CTSK P43235 11/20 0.42
CTSS P25774 5/20 0.42
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
KMT2A Q03164 1/20 0.40
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CA12 O43570 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA4 P22748 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14923533 1.00 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL22383165 1.00 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL13617298 1.00 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL17564382 1.00 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL14923484 1.00 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL14923728 1.00 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL24069882 0.87 CA1 (0.57) CA1CA2CA7CYP2D6CTSK
SCHEMBL14842451 0.86 CA1 (0.49) CA1CA2CA7CYP2D6CTSK
SCHEMBL15081449 0.84 CA1 (0.51) CA1CA2CA7CYP2D6CTSK
SCHEMBL12396266 0.83 CA1 (0.58) CA1CA2CA7CYP2D6CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed
EP-2589592-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM Corporation (JP) 2013-05-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, CD38, BTK CA1 3179/4885CA2 688/4885CA7 2926/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.