SCHEMBL14939381

SCHEMBL14939381

O=C1c2ccccc2CC1(c1ccccc1)N1CCN(Cc2ccncc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.54
SIGMAR1 Q99720 5/20 0.46
DRD2 P14416 3/20 0.46
HTR2A P28223 3/20 0.46
HTR2C P28335 3/20 0.46
HTR2B P41595 3/20 0.46
OPRL1 P41146 1/20 0.45
TSHR P16473 3/20 0.43
KDM4E B2RXH2 2/20 0.43
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
USP2 O75604 1/20 0.41
TP53 P04637 1/20 0.41
CCR2 P41597 1/20 0.41
MC4R P32245 1/20 0.40
TRPV6 Q9H1D0 1/20 0.40
KDM1A O60341 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939625 0.92 NPSR1 (0.64) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939175 0.92 NPSR1 (0.64) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14940373 0.92 NPSR1 (0.64) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14940132 0.88 NPSR1 (0.51) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939037 0.87 NPSR1 (0.58) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939177 0.84 NPSR1 (0.54) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939931 0.83 KMT2A (0.48) NPSR1SIGMAR1OPRL1TSHRKDM4E
SCHEMBL14938983 0.82 NPSR1 (0.55) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939777 0.81 NPSR1 (0.54) NPSR1SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939466 0.81 NPSR1 (0.54) NPSR1SIGMAR1DRD2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed