SCHEMBL14939436

SCHEMBL14939436

COc1cccc(CN2CCN(C3(c4ccccc4)C(=O)c4cccc(Cl)c4C3=O)CC2)c1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.61
SIGMAR1 Q99720 1/20 0.57
TSHR P16473 2/20 0.52
GAA P10253 1/20 0.52
ALDH1A1 P00352 3/20 0.48
ALDH3A1 P30838 1/20 0.48
MAPT P10636 3/20 0.48
CHRM2 P08172 1/20 0.47
CHRM3 P20309 1/20 0.47
MMP2 P08253 2/20 0.46
MMP9 P14780 2/20 0.46
FAAH O00519 1/20 0.46
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
KDM4E B2RXH2 2/20 0.45
LMNA P02545 2/20 0.45
RECQL P46063 1/20 0.45
ATM Q13315 1/20 0.44
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940106 0.90 NPSR1 (0.72) NPSR1SIGMAR1GAAALDH1A1ALDH3A1
SCHEMBL14939022 0.90 NPSR1 (0.59) NPSR1SIGMAR1ALDH1A1ALDH3A1MAPT
SCHEMBL14939688 0.89 NPSR1 (0.77) NPSR1SIGMAR1MAPTMMP2MMP9
SCHEMBL14939350 0.89 NPSR1 (0.58) NPSR1SIGMAR1ALDH1A1ALDH3A1MAPT
SCHEMBL14939441 0.88 NPSR1 (0.72) NPSR1SIGMAR1ALDH1A1ALDH3A1MAPT
SCHEMBL14939713 0.88 NPSR1 (0.65) NPSR1SIGMAR1TSHRGAAALDH1A1
SCHEMBL14939979 0.85 NPSR1 (0.61) NPSR1SIGMAR1TSHRGAAALDH1A1
SCHEMBL14939758 0.85 NPSR1 (0.63) NPSR1SIGMAR1TSHRGAAALDH1A1
SCHEMBL14939975 0.84 NPSR1 (0.60) NPSR1SIGMAR1TSHRGAAALDH1A1
SCHEMBL14939475 0.83 NPSR1 (0.58) NPSR1SIGMAR1TSHRGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed