SCHEMBL1494701

SCHEMBL1494701

COc1ccn(-c2ccccc2)c1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.49
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43
TUBA1A Q71U36 1/20 0.43
TUBA1C Q9BQE3 1/20 0.43
TUBB6 Q9BUF5 1/20 0.43
TUBB2B Q9BVA1 1/20 0.43
TUBB1 Q9H4B7 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15506073 0.79 CA12 (0.51) NOTUMCA12CA1CA2CA7
SCHEMBL11453643 0.74 NOTUM (0.65) NOTUMCA12CA1CA2CA7
SCHEMBL5153925 0.74 CA1 (0.44) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL29626125 0.73 CA12 (0.41) NOTUMCA12CA1CA2CA7
SCHEMBL12998009 0.73 NOTUM (0.49) NOTUMALDH1A1HPGDKDM4EFGFR1
SCHEMBL3264191 0.72 NOTUM (0.62) NOTUMALDH1A1HPGDKDM4EHTT
SCHEMBL4980499 0.71 NOTUM (0.47) NOTUMKDM4ECOMTMAPTPOLB
SCHEMBL732887 0.71 CA12 (0.45) NOTUMTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL10059740 0.68 GAA (0.46) CA12CA1CA2CA7CA9
SCHEMBL16031477 0.68 MEN1 (0.44) NOTUMALDH1A1HPGDKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2475660-A1 PYRROLO-PYRIDINE DERIVATIVES AS ACTIVATORS OF AMPK GlaxoSmithKline LLC (US) 2012-07-18 EP disclosed
WO-2011029855-A1 PYRROLO-PYRIDINE DERIVATIVES AS ACTIVATORS OF AMPK GLAXOSMITHKLINE LLC (US) 2011-03-17 WO disclosed