SCHEMBL14949374

SCHEMBL14949374

COc1ccc2c(Oc3cc(-c4nnc(Nc5cccc(C)c5)[nH]4)ccc3C)ccnc2c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.42
PDGFRA P16234 2/20 0.42
MET P08581 7/20 0.42
FGFR2 P21802 3/20 0.38
TEK Q02763 3/20 0.38
AURKA O14965 2/20 0.38
AURKB Q96GD4 1/20 0.38
AXL P30530 1/20 0.38
LCK P06239 1/20 0.37
TLR8 Q9NR97 1/20 0.37
GAK O14976 1/20 0.37
RIPK2 O43353 1/20 0.37
COQ8A Q8NI60 1/20 0.37
NLK Q9UBE8 1/20 0.37
EGFR P00533 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14949214 0.91 KDR (0.49) KDRPDGFRAMETFGFR2TEK
SCHEMBL14949313 0.90 KDR (0.46) KDRPDGFRAMETFGFR2TEK
SCHEMBL12336455 0.90 GSK3A (0.47) KDRMETAXLGAKEGFR
SCHEMBL14949221 0.86 FGFR2 (0.49) KDRPDGFRAMETFGFR2TEK
SCHEMBL14949208 0.85 KDR (0.46) KDRPDGFRAMETFGFR2TEK
SCHEMBL14949223 0.84 KDR (0.49) KDRPDGFRAMETFGFR2TEK
SCHEMBL14949353 0.83 KDR (0.45) KDRPDGFRAMETFGFR2TEK
SCHEMBL16786015 0.82 KDR (0.60) KDRPDGFRAMETFGFR2TEK
SCHEMBL14949367 0.82 KDR (0.42) KDRPDGFRAMETFGFR2TEK
SCHEMBL14949232 0.82 KDR (0.46) KDRPDGFRAMETFGFR2AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160096824-A1 Heterocyclic Compounds Useful for Kinase Inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. 2016-04-07 US disclosed
US-9212151-B2 Heterocyclic compounds useful for kinase inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. (US) 2015-12-15 US disclosed
US-20150158828-A1 Heterocyclic Compounds Useful for Kinase Inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. 2015-06-11 US disclosed
US-8957216-B2 Heterocyclic compounds useful for kinase inhibition AMITECH THERAPEUTIC SOLUTIONS, INC. (US) 2015-02-17 US disclosed
US-20130123284-A1 HETEROCYCLIC COMPOUNDS USEFUL FOR KINASE INHIBITION AMITECH THERAPEUTIC SOLUTIONS INC (US) 2013-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123284-A1 HETEROCYCLIC COMPOUNDS USEFUL FOR KINASE INHIBITION MAP4K2, MAP3K20, MAP3K19 KDR 533/4885PDGFRA 498/4885MET 770/4885
US-20150158828-A1 Heterocyclic Compounds Useful for Kinase Inhibition MAP4K2, MAP3K20, MAP3K19 KDR 533/4885PDGFRA 498/4885MET 770/4885
US-20160096824-A1 Heterocyclic Compounds Useful for Kinase Inhibition MAP4K2, MAP3K20, MAP3K19 KDR 533/4885PDGFRA 498/4885MET 770/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.