SCHEMBL14958754

SCHEMBL14958754

COc1cc(C)c(S(=O)(=O)N(C)CCC(=O)Nc2ccc(N3CCCCC3)cc2)c(C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.54
TP53 P04637 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
KMT2A Q03164 5/20 0.51
ALDH1A1 P00352 5/20 0.51
USP2 O75604 3/20 0.51
KDM4E B2RXH2 3/20 0.51
ALOX15 P16050 2/20 0.51
NR4A1 P22736 2/20 0.51
MCL1 Q07820 2/20 0.51
MAPK1 P28482 2/20 0.51
BDKRB1 P46663 1/20 0.50
MEN1 O00255 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP3A4 P08684 1/20 0.49
PTK2B Q14289 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3439838 0.92 MAPT (0.49) MAPTTP53SMN1; SMN2KMT2AALDH1A1
SCHEMBL3440040 0.92 BDKRB1 (0.53) MAPTSMN1; SMN2RAB9ANPC1KMT2A
SCHEMBL3440208 0.92 BDKRB1 (0.54) MAPTKMT2AALDH1A1USP2KDM4E
SCHEMBL12912382 0.91 BDKRB1 (0.49) MAPTSMN1; SMN2KMT2AALDH1A1USP2
SCHEMBL3439617 0.90 BDKRB1 (0.48) MAPTSMN1; SMN2KMT2AALDH1A1USP2
SCHEMBL12914508 0.90 POLB (0.55) MAPTSMN1; SMN2RAB9ANPC1KMT2A
SCHEMBL3439589 0.90 BDKRB1 (0.49) MAPTKMT2AALDH1A1USP2KDM4E
SCHEMBL3440534 0.89 BDKRB1 (0.47) MAPTSMN1; SMN2KMT2AALDH1A1USP2
SCHEMBL3440280 0.89 BDKRB1 (0.51) MAPTMAPK1BDKRB1LMNA
SCHEMBL3440009 0.89 BDKRB1 (0.51) MAPTMAPK1BDKRB1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402329-B1 Analgetic phenylsulphonamides BOEHRINGER INGELHEIM INT (DE) 2013-05-22 EP disclosed