SCHEMBL1496052

SCHEMBL1496052

Cc1ccc2c(c1)Nc1c(cnn1C)CN2C(=O)C1CCC(CNC(=O)C2CCN(CC3CC3)CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 13/20 0.39
KMT2A Q03164 1/20 0.38
IDH1 O75874 2/20 0.38
OXTR P30559 7/20 0.38
AVPR2 P30518 3/20 0.37
ACKR3 P25106 1/20 0.37
EPHX2 P34913 1/20 0.37
WNT1 P04628 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1496007 0.94 AVPR1A (0.42) AVPR1AIDH1OXTRAVPR2
SCHEMBL1496255 0.92 IDH1 (0.38) AVPR1AIDH1OXTRAVPR2WNT1
SCHEMBL1496081 0.90 AVPR1A (0.45) AVPR1AOXTRAVPR2
SCHEMBL1495943 0.90 IDH1 (0.46) AVPR1AIDH1OXTR
SCHEMBL1495996 0.88 AVPR1A (0.45) AVPR1AOXTRAVPR2
SCHEMBL1495930 0.85 AVPR1A (0.40) AVPR1AIDH1OXTRAVPR2
SCHEMBL18944285 0.85 AVPR1A (0.40) AVPR1AIDH1OXTRAVPR2
SCHEMBL2628963 0.84 AVPR1A (0.41) AVPR1AIDH1OXTRAVPR2
SCHEMBL12832107 0.84 AVPR1A (0.40) AVPR1AIDH1OXTRAVPR2
SCHEMBL12832110 0.83 IDH1 (0.48) AVPR1AIDH1OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2292621-A1 Vasopressin v1a antagonists Vantia Limited (GB) 2011-03-09 EP claimed