SCHEMBL1496070

SCHEMBL1496070

Cn1ncc2c1Nc1ccccc1N(C(=O)C1CCC(CNC(=O)N3CCN(CCC(C)(C)C)CC3)CC1)C2

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 18/20 0.49
OXTR P30559 7/20 0.49
AVPR2 P30518 2/20 0.49
IDH1 O75874 2/20 0.44
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM3 P20309 1/20 0.43
DRD3 P35462 1/20 0.43
OPRK1 P41145 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1496002 0.91 AVPR1A (0.52) AVPR1AOXTRAVPR2IDH1CHRM2
SCHEMBL1496024 0.91 AVPR1A (0.43) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL1495887 0.90 AVPR1A (0.45) AVPR1AOXTRIDH1
SCHEMBL1496011 0.90 AVPR1A (0.41) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL1496146 0.84 AVPR1A (0.43) AVPR1AOXTRAVPR2IDH1CHRM2
SCHEMBL1495998 0.83 IDH1 (0.52) AVPR1AOXTRAVPR2IDH1
SCHEMBL1496103 0.82 AVPR1A (0.44) AVPR1AOXTRAVPR2IDH1CHRM2
SCHEMBL1496069 0.81 AVPR1A (0.42) AVPR1AOXTRAVPR2IDH1CHRM2
SCHEMBL2631708 0.81 IDH1 (0.47) AVPR1AOXTRAVPR2IDH1
SCHEMBL1496081 0.81 AVPR1A (0.45) AVPR1AOXTRAVPR2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2292621-A1 Vasopressin v1a antagonists Vantia Limited (GB) 2011-03-09 EP claimed