SCHEMBL14964355

SCHEMBL14964355

CC(C)(C)OC(=O)N1CCC(C)(C(=O)Nc2cccc(Oc3ccc(F)cc3)c2)CC1.CC(C)(C)OC(=O)N1CCC(C)(C(=O)O)CC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 9/20 0.50
HDAC2 Q92769 2/20 0.45
HDAC1 Q13547 1/20 0.45
OTUD7B Q6GQQ9 1/20 0.44
USP2 O75604 2/20 0.43
CYP3A4 P08684 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP2C9 P11712 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP1A2 P05177 2/20 0.42
NTRK1 P04629 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
MET P08581 1/20 0.41
AXL P30530 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4290419 0.97 S1PR2 (0.52) S1PR2HDAC2HDAC1OTUD7BUSP2
SCHEMBL1446881 0.86 S1PR2 (0.56) S1PR2OTUD7BUSP2CYP3A4ALDH1A1
SCHEMBL20137661 0.81 TSHR (0.52) CYP3A4ALDH1A1CYP1A2CYP2C19
SCHEMBL1447574 0.80 LIMK2 (0.55) EPHX2
SCHEMBL4866877 0.80 PTPN2 (0.59) S1PR2ALDH1A1
SCHEMBL1446944 0.77 S1PR2 (0.48) S1PR2OTUD7BUSP2ALDH1A1SMN1; SMN2
SCHEMBL1446961 0.77 CA1 (0.50) ALDH1A1
SCHEMBL31058161 0.77 ANO1 (0.53) S1PR2EPHX2
SCHEMBL31058254 0.76 PARP14 (0.49) EPHX2
SCHEMBL20137885 0.76 TSHR (0.44) HDAC2HDAC1NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8450332-B2 LIMK2 inhibitors, compositions comprising them, and methods of their use LEXICON PHARMACEUTICALS, INC. (US) 2013-05-28 US disclosed