SCHEMBL14967335

SCHEMBL14967335

Cc1cc(C)c(CNC(=O)c2ccc([C@@H](C)c3ccccc3)cc2)c(O)n1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 6/20 0.48
SMN1; SMN2 Q16637 3/20 0.43
HPGD P15428 2/20 0.42
HSD17B10 Q99714 1/20 0.42
ALDH1A1 P00352 3/20 0.42
RAB9A P51151 1/20 0.42
TP53 P04637 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
LMNA P02545 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PKM P14618 1/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14967167 1.00 KLKB1 (0.48) KLKB1SMN1; SMN2HPGDHSD17B10ALDH1A1
SCHEMBL14967617 1.00 KLKB1 (0.48) KLKB1SMN1; SMN2HPGDHSD17B10ALDH1A1
SCHEMBL14966917 0.90 KLKB1 (0.44) KLKB1SMN1; SMN2HPGDALDH1A1OPRM1
SCHEMBL14966902 0.90 KLKB1 (0.44) KLKB1SMN1; SMN2HPGDALDH1A1OPRM1
SCHEMBL14972066 0.90 KLKB1 (0.44) KLKB1SMN1; SMN2HPGDALDH1A1OPRM1
SCHEMBL14966450 0.88 SMN1; SMN2 (0.46) KLKB1SMN1; SMN2HPGDHSD17B10ALDH1A1
SCHEMBL17319363 0.88 KLKB1 (0.43) KLKB1SMN1; SMN2ALDH1A1OPRM1OPRK1
SCHEMBL17319364 0.88 KLKB1 (0.43) KLKB1SMN1; SMN2ALDH1A1OPRM1OPRK1
SCHEMBL14966658 0.87 SMN1; SMN2 (0.45) KLKB1SMN1; SMN2HPGDHSD17B10ALDH1A1
SCHEMBL14967419 0.87 SMN1; SMN2 (0.45) KLKB1SMN1; SMN2HPGDHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780014-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF Constellation Pharmaceuticals, Inc. (US) 2014-09-24 EP disclosed
WO-2013075083-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed