SCHEMBL14972809

SCHEMBL14972809

O=C1OCCCC1=CO.[NaH]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.47
DYRK1A Q13627 6/20 0.44
DYRK1B Q9Y463 6/20 0.44
CLK1 P49759 2/20 0.44
MAPT P10636 3/20 0.42
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
ALOX5 P09917 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
DYRK2 Q92630 3/20 0.32
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28943338 1.00 NAMPT (0.47) NAMPTDYRK1ADYRK1BCLK1MAPT
SCHEMBL9686981 0.98
SCHEMBL9686986 0.98
SCHEMBL29597368 0.96 NAMPT (0.47) NAMPTDYRK1ADYRK1BCLK1MAPT
SCHEMBL1311913 0.86
SCHEMBL2834476 0.84
SCHEMBL3972493 0.84
SCHEMBL9943877 0.84
SCHEMBL980488 0.76
SCHEMBL30881494 0.74 NAMPT (0.47) NAMPTDYRK1ADYRK1BCLK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391614-B1 ENAMINOCARBONYL COMPOUNDS AND THEIR USE INST CHEMII ORGANICZNEJ POLSKA AKADEMIA NAUK (PL) 2013-05-29 EP disclosed