SCHEMBL1497367

SCHEMBL1497367

CC(=O)C=C(C)CN1CCN(C2CCN(c3cc(-c4cnc(N)nc4)nc(N4CCOCC4)c3)CC2)CC1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 0.49
AKT1 P31749 14/20 0.49
MTOR P42345 9/20 0.49
MAP3K12 Q12852 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2396675 0.91 PIK3CA (0.50) PIK3CAAKT1MTORMAP3K12
SCHEMBL1497656 0.83 PIK3CA (0.50) PIK3CAAKT1MTORMAP3K12
SCHEMBL1309681 0.76 PIK3CA (0.71) PIK3CAAKT1MTORMAP3K12
SCHEMBL12264937 0.74 PIK3CA (0.47) PIK3CAAKT1MTORMAP3K12
SCHEMBL27935452 0.72 PIK3CA (0.61) PIK3CAAKT1MTORMAP3K12
SCHEMBL13174417 0.72 PIK3CA (0.65) PIK3CAAKT1MTORMAP3K12
SCHEMBL1497654 0.72 PIK3CA (0.47) PIK3CAAKT1MTORMAP3K12
SCHEMBL2393055 0.71 PIK3CA (0.51) PIK3CAAKT1MTORMAP3K12
SCHEMBL1497596 0.69 PIK3CA (0.45) PIK3CAAKT1MTORMAP3K12
SCHEMBL12488973 0.69 PIK3CA (0.57) PIK3CAAKT1MTORMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2475375-A2 PI3 KINASE INHIBITORS AND USES THEREOF Avila Therapeutics, Inc. (US) 2012-07-18 EP disclosed
WO-2011031896-A2 PI3 KINASE INHIBITORS AND USES THEREOF AVILA THERAPEUTICS, INC. (US) 2011-03-17 WO disclosed